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1

Influence of formulation composition and process on the characteristics and in vitro release from PLGA-based sustained release injectables

Meeus, Joke, Scurr, David J., Appeltans, Bernard, Amssoms, Katie, Annaert, Pieter, Davies, Martyn C., Roberts, Clive J., Van den Mooter, Guy

Journal:

European Journal of Pharmaceutics and Biopharmaceutics

Year:

2015

Language:

english

File:

PDF, 2.12 MB

english, 2015

2

Design and Optimization of Tricyclic Phtalimide Analogues as Novel Inhibitors of HIV-1 Integrase

Verschueren, Wim G., Dierynck, Inge, Amssoms, Katie I. E., Hu, Lili, Boonants, Paul M. J. G., Pille, Geert M. E., Daeyaert, Frits F. D., Hertogs, Kurt, Surleraux, Dominique L. N. G., Wigerinck, Piet B

Journal:

Journal of Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 322 KB

english, 2005

3

ChemInform Abstract: An Efficient Synthesis of Orthogonally Protected Spermidine.

K. Amssoms, K. Augustyns, A. Yamani, M. Zhang, A. Haemers

Journal:

Year:

2002

File:

PDF, 30 KB

2002

4

1,5-Benzodiazepine inhibitors of HCV NS5B polymerase

David McGowan, Origène Nyanguile, Maxwell D. Cummings, Sandrine Vendeville, Koen Vandyck, Walter Van den Broeck, Carlo W. Boutton, Hendrik De Bondt, Ludo Quirynen, Katie Amssoms, Jean-François Bonfant

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 1.04 MB

english, 2009

5

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 1: Substitution of the glycine carboxylic acid group

Katie Amssoms, Sandra L Oza, Esteban Ravaschino, Abdellah Yamani, Anne-Marie Lambeir, Padinchare Rajan, Gunther Bal, Juan Bautista Rodriguez, Alan H Fairlamb, Koen Augustyns, Achiel Haemers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 115 KB

english, 2002

6

Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: Substitution of the glycine part

Katie Amssoms, Sandra L Oza, Koen Augustyns, Abdellah Yamani, Anne-Marie Lambeir, Gunther Bal, Pieter Van der Veken, Alan H Fairlamb, Achiel Haemers

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 95 KB

english, 2002

7

Structure-Based Macrocyclization Yields Hepatitis C Virus NS5B Inhibitors with Improved Binding Affinities and Pharmacokinetic Properties

Dr. Maxwell D. Cummings, Dr. Tse-I Lin, Lili Hu, Dr. Abdellah Tahri, David McGowan, Dr. Katie Amssoms, Stefaan Last, Dr. Benoit Devogelaere, Marie-Claude Rouan, Dr. Leen Vijgen, Dr. Jan Martin Berke,

Journal:

Angewandte Chemie

Year:

2012

Language:

english

File:

PDF, 713 KB

english, 2012

8

Structure-Based Macrocyclization Yields Hepatitis C Virus NS5B Inhibitors with Improved Binding Affinities and Pharmacokinetic Properties

Dr. Maxwell D. Cummings, Dr. Tse-I Lin, Lili Hu, Dr. Abdellah Tahri, David McGowan, Dr. Katie Amssoms, Stefaan Last, Dr. Benoit Devogelaere, Marie-Claude Rouan, Dr. Leen Vijgen, Dr. Jan Martin Berke,

Journal:

Angewandte Chemie International Edition

Year:

2012

Language:

english

File:

PDF, 720 KB

english, 2012

9

Nanoscale surface characterization and miscibility study of a spray-dried injectable polymeric matrix consisting of poly(lactic-co-glycolic acid) and polyvinylpyrrolidone

Joke Meeus, Xinyong Chen, David J. Scurr, Valeria Ciarnelli, Katie Amssoms, Clive J. Roberts, Martyn C. Davies, Guy van Den Mooter

Journal:

Journal of Pharmaceutical Sciences

Year:

2012

Language:

english

File:

PDF, 584 KB

english, 2012

10

Finger loop inhibitors of the HCV NS5b polymerase. Part II. Optimization of tetracyclic indole-based macrocycle leading to the discovery of TMC647055

Sandrine Vendeville, Tse-I. Lin, Lili Hu, Abdellah Tahri, David McGowan, Maxwell D. Cummings, Katie Amssoms, Maxime Canard, Stefaan Last, Iris Van den Steen, Benoit Devogelaere, Marie-Claude Rouan, Le

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 1.62 MB

english, 2012

11

Finger-loop inhibitors of the HCV NS5b polymerase. Part 1: Discovery and optimization of novel 1,6- and 2,6-macrocyclic indole series

David McGowan, Sandrine Vendeville, Tse-I Lin, Abdellah Tahri, Lili Hu, Maxwell D. Cummings, Katie Amssoms, Jan Martin Berke, Maxime Canard, Erna Cleiren, Pascale Dehertogh, Stefaan Last, Els Fransen,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 1.38 MB

english, 2012

12

Structure-Based Design of a Benzodiazepine Scaffold Yields a Potent Allosteric Inhibitor of Hepatitis C NS5B RNA Polymerase

Vandyck, Koen, Cummings, Maxwell D., Nyanguile, Origène, Boutton, Carlo W., Vendeville, Sandrine, McGowan, David, Devogelaere, Benoit, Amssoms, Katie, Last, Stefaan, Rombauts, Klara, Tahri, Abdellah,

Journal:

Journal of Medicinal Chemistry

Year:

2009

Language:

english

File:

PDF, 2.11 MB

english, 2009

13

Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application

Kesteleyn, Bart, Amssoms, Katie, Schepens, Wim, Hache, Geerwin, Verschueren, Wim, Van De Vreken, Wim, Rombauts, Klara, Meurs, Greet, Sterkens, Patrick, Stoops, Bart, Baert, Lieven, Austin, Nigel, Wegn

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 1.32 MB

english, 2013

14

Discovery and Early Development of TMC647055, a Non-Nucleoside Inhibitor of the Hepatitis C Virus NS5B Polymerase

Cummings, Maxwell D., Lin, Tse-I, Hu, Lili, Tahri, Abdellah, McGowan, David, Amssoms, Katie, Last, Stefaan, Devogelaere, Benoit, Rouan, Marie-Claude, Vijgen, Leen, Berke, Jan Martin, Dehertogh, Pascal

Journal:

Journal of Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 2.90 MB

english, 2014

15

Surface Characteristics of Spray-Dried Microspheres Consisting of PLGA and PVP: Relating the Influence of Heat and Humidity to the Thermal Characteristics of These Polymers

Meeus, Joke, Scurr, David J., Amssoms, Katie, Davies, Martyn C., Roberts, Clive J., Van den Mooter, Guy

Journal:

Molecular Pharmaceutics

Year:

2013

Language:

english

File:

PDF, 2.17 MB

english, 2013

16

TMC647055, a Potent Nonnucleoside Hepatitis C Virus NS5B Polymerase Inhibitor with Cross-Genotypic Coverage

Devogelaere, B., Berke, J. M., Vijgen, L., Dehertogh, P., Fransen, E., Cleiren, E., van der Helm, L., Nyanguile, O., Tahri, A., Amssoms, K., Lenz, O., Cummings, M. D., Clayton, R. F., Vendeville, S.,

Journal:

Antimicrobial Agents and Chemotherapy

Year:

2012

Language:

english

File:

PDF, 703 KB

english, 2012

17

Trypanothione as a Target in the Design of Antitrypanosomal and Antileishmanial Agents

Augustyns, K., Amssoms, K., Yamani, A., Rajan, P., Haemers, A.

Journal:

Current Pharmaceutical Design

Year:

2001

Language:

english

File:

PDF, 123 KB

english, 2001

18

AN EFFICIENT SYNTHESIS OF ORTHOGONALLY PROTECTED SPERMIDINE

Amssoms, K., Augustyns, K., Yamani, A., Zhang, M., Haemers, A.

Journal:

Synthetic Communications

Year:

2002

Language:

english

File:

PDF, 138 KB

english, 2002

19

In vivo evaluation of different formulation strategies for sustained release injectables of a poorly soluble HIV protease inhibitor

Meeus, Joke, Scurr, David J., Amssoms, Katie, Wuyts, Koen, Annaert, Pieter, Davies, Martyn C., Roberts, Clive J., Van den Mooter, Guy

Journal:

Journal of Controlled Release

Year:

2015

Language:

english

File:

PDF, 1.33 MB

english, 2015

20

The Influence of Spray-Drying Parameters on Phase Behavior, Drug Distribution, and In Vitro Release of Injectable Microspheres for Sustained Release

Meeus, Joke, Lenaerts, Maité, Scurr, David J., Amssoms, Katie, Davies, Martyn C., Roberts, Clive J., Van Den Mooter, Guy

Journal:

Journal of Pharmaceutical Sciences

Year:

2015

Language:

english

File:

PDF, 704 KB

english, 2015

21

Combination of (M)DSC and Surface Analysis to Study the Phase Behaviour and Drug Distribution of Ternary Solid Dispersions

Meeus, Joke, Scurr, David J., Chen, Xinyong, Amssoms, Katie, Davies, Martyn C., Roberts, Clive J., Van den Mooter, Guy

Journal:

Pharmaceutical Research

Year:

2015

Language:

english

File:

PDF, 4.14 MB

english, 2015

22

Sustained release of the candidate antiretroviral peptides T-1249 and JNJ54310516-AFP from a rod insert vaginal ring

Murphy, Diarmaid J., Amssoms, Katie, Pille, Geert, Clarke, Aileen, O’Hara, Marc, van Roey, Jens, Malcolm, R. Karl

Journal:

Drug Delivery and Translational Research

Year:

2016

Language:

english

File:

PDF, 802 KB

english, 2016

23

Humanized Mice Recapitulate Key Features of HIV-1 Infection: A Novel Concept Using Long-Acting Anti-Retroviral Drugs for Treating HIV-1

Nischang, Marc, Sutmuller, Roger, Gers-Huber, Gustavo, Audigé, Annette, Li, Duo, Rochat, Mary-Aude, Baenziger, Stefan, Hofer, Ursula, Schlaepfer, Erika, Regenass, Stephan, Amssoms, Katie, Stoops, Bart

Journal:

Year:

2012

Language:

english

File:

PDF, 1.12 MB

english, 2012

24

2,4-Diaminoquinazolines as Dual Toll Like Receptor (TLR) 7/8 Modulators for the Treatment of Hepatitis B Virus

Embrechts, Werner, Herschke, Florence, Pauwels, Frederik, Stoops, Bart, Last, Stefaan, Pieters, Serge, Pande, Vineet, Pille, Geert, Amssoms, Katie, Smyej, Ilham, Dhuyvetter, Deborah, Scholliers, Annic

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 1.81 MB

english, 2018

25

Ovalbumin-containing core-shell implants suitable to obtain a delayed IgG1 antibody response in support of a biphasic pulsatile release profile in mice

Amssoms, Katie, Born, Philip A., Beugeling, Max, De Clerck, Ben, Van Gulck, Ellen, Hinrichs, Wouter L. J., Frijlink, Henderik W., Grasmeijer, Niels, Kraus, Guenter, Sutmuller, Roger, Simmen, Kenny, Ba

Journal:

Year:

2018

Language:

english

File:

PDF, 3.57 MB

english, 2018

26

The mechanism behind the biphasic pulsatile drug release from physically mixed poly(dl-lactic(-co-glycolic) acid)-based compacts

Beugeling, Max, Grasmeijer, Niels, Born, Philip A., van der Meulen, Merel, van der Kooij, Renée S., Schwengle, Kevin, Baert, Lieven, Amssoms, Katie, Frijlink, Henderik W., Hinrichs, Wouter L.J.

Journal:

International Journal of Pharmaceutics

Year:

2018

Language:

english

File:

PDF, 1.21 MB

english, 2018

27

DISCOVERY OF A NOVEL, POTENTIAL FIRST-IN-CLASS MALT1 PROTEASE INHIBITOR FOR THE TREATMENT OF B CELL LYMPHOMAS

Philippar, U., Lu, T., Vloemans, N., Bekkers, M., van Nuffel, L., Gaudiano, M., Wnuk-Lipinska, K., Van Der Leede, B., Amssoms, K., Kimpe, K., Medaer, B., Greway, T., Abraham, Y., Cummings, M., Trella,

Journal:

Hematological Oncology

Year:

2019

Language:

english

File:

PDF, 106 KB

english, 2019

28

DISCOVERY OF A NOVEL, POTENTIAL FIRST-IN-CLASS MALT1 PROTEASE INHIBITOR FOR THE TREATMENT OF B CELL LYMPHOMAS

Philippar, U., Lu, T., Vloemans, N., Bekkers, M., van Nuffel, L., Gaudiano, M., Wnuk-Lipinska, K., Van Der Leede, B., Amssoms, K., Kimpe, K., Medaer, B., Greway, T., Abraham, Y., Cummings, M., Trella,

Journal:

Hematological Oncology

Year:

2019

File:

PDF, 106 KB

2019

29

Development of a Stable Respiratory Syncytial Virus Pre-Fusion Protein Powder Suitable for a Core-Shell Implant with a Delayed Release in Mice: A Proof of Concept Study

Beugeling,, Amssoms,, Cox,, De Clerck,, Van Gulck,, Verwoerd,, Kraus,, Roymans,, Baert,, Frijlink,, Hinrichs,

Journal:

Year:

2019

File:

PDF, 856 KB

2019

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